G-protein coupled receptors (GPCRs) form the largest class of cell-surface receptors. There are ~ 800 GPCRs overall, and as such this target class is very important in drug discovery. Currently around, ~ 35% of all drugs approved by the FDA act at 108 unique GPCRs1.
Customized assays are routinely provided by scientific teams upon request.
Radioligand binding and functional assays (Read More for Targets and Assays)